5-HT1F receptor

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Lua error in Module:Infobox_gene at line 33: attempt to index field 'wikibase' (a nil value). 5-hydroxytryptamine (serotonin) receptor 1F, also known as HTR1F is a 5-HT1 receptor protein and also denotes the human gene encoding it.[1][2][3][4][5]

Agonists

  • 5-n-Butyryloxy-DMT:[6] >60-fold selectivity versus 5-HT1E receptor
  • BRL-54443 - mixed 5-HT1E/1F agonist
  • Eletriptan - mixed 5-HT1B/1D/1E/1F/2B/7 agonist
  • LY-334,370[7] - as well as related benzamides[8]
  • LY-344,864 (N-[(3R)-3-(Dimethylamino)-2,3,4,9-tetrahydro-1H-carbazol-6-yl]-4-fluorobenzamide)
  • Naratriptan - mixed 5-HT1B/1D/1F agonist

Antagonists

MLS000756415[9]

See also

References

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  9. PudChem: MLS000756415

Further reading

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External links

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This article incorporates text from the United States National Library of Medicine, which is in the public domain.



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