Cinolazepam

From Infogalactic: the planetary knowledge core
Jump to: navigation, search

<templatestyles src="Module:Hatnote/styles.css"></templatestyles>

Cinolazepam
Cinolazepam.svg
Cinolazepam3d.png
Systematic (IUPAC) name
(RS)-3-[9-Chloro-6-(2-fluorophenyl)-4-hydroxy-3-oxo-2,5-diazabicyclo[5.4.0]undeca-5,8,10,12-tetraen-2-yl]propanenitrile
Clinical data
Trade names Gerodorm
AHFS/Drugs.com International Drug Names
Pregnancy
category
  •  ?
Legal status
Routes of
administration
Oral
Pharmacokinetic data
Bioavailability 90–100%
Metabolism Hepatic
Biological half-life 9 hours[1]
Excretion Renal
Identifiers
CAS Number 75696-02-5 YesY
ATC code N05CD13 (WHO)
PubChem CID: 3033621
DrugBank DB01594 YesY
ChemSpider 2298251 YesY
UNII 68P0556B0U YesY
KEGG D07328 YesY
ChEBI CHEBI:59514 YesY
ChEMBL CHEMBL2104926 N
Chemical data
Formula C18H13ClFN3O2
Molecular mass 357.8
  • FC1=CC=CC=C1C2=NC(C(N(CCC#N)C3=C2C=C(C=C3)Cl)=O)O
  • InChI=1S/C18H13ClFN3O2/c19-11-6-7-15-13(10-11)16(12-4-1-2-5-14(12)20)22-17(24)18(25)23(15)9-3-8-21/h1-2,4-7,10,17,24H,3,9H2 YesY
  • Key:XAXMYHMKTCNRRZ-UHFFFAOYSA-N YesY
 NYesY (what is this?)  (verify)

Cinolazepam[2] (marketed under the brand name Gerodorm)[3] is a drug which is a benzodiazepine derivative. It possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. Due to its strong sedative properties, it is primarily used as an hypnotic.

Cinolazepam is not approved for sale in the United States or Canada.

See also

References

  1. Lua error in package.lua at line 80: module 'strict' not found.
  2. US Patent 4388313 Novel 3-hydroxy-1,4-benzodiazepine-2-ones and process for the preparation thereof
  3. Lua error in package.lua at line 80: module 'strict' not found.

External links

<templatestyles src="Asbox/styles.css"></templatestyles>