Imagabalin

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Imagabalin
Imagabalin.svg
Systematic (IUPAC) name
(3S,5R)-3-amino-5-methyloctanoic acid
Identifiers
CAS Number 610300-07-7
610300-00-0 (hydrochloride)
ATC code None
PubChem CID: 10236037
ChemSpider 8411525
Synonyms PD-0332334; PD-332,334
Chemical data
Formula C9H19NO2
Molecular mass 173.253 g/mol
  • O=C(O)C[C@@H](N)C[C@@H](CCC)C
  • InChI=1S/C9H19NO2/c1-3-4-7(2)5-8(10)6-9(11)12/h7-8H,3-6,10H2,1-2H3,(H,11,12)/t7-,8+/m1/s1
  • Key:JXEHXYFSIOYTAH-SFYZADRCSA-N

Imagabalin (INN, USAN; PD-332,334) is a drug which acts as a ligand for the α2δ subunit of the voltage-dependent calcium channel,[1] with some selectivity for the α2δ1 subunit over α2δ2.[2] Under development by Pfizer as a pharmaceutical medication, it has demonstrated preclinical efficacy of anxiolytic, analgesic, hypnotic, and anticonvulsant-like activity and is currently in phase III clinical trials for the treatment of generalized anxiety disorder.[2][3]

See also

References

  1. ↑ Lua error in package.lua at line 80: module 'strict' not found.
  2. ↑ 2.0 2.1 Lua error in package.lua at line 80: module 'strict' not found.
  3. ↑ Lua error in package.lua at line 80: module 'strict' not found.


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