Bromadoline
From Infogalactic: the planetary knowledge core
![]() |
|
Systematic (IUPAC) name | |
---|---|
trans-4-bromo-N-(2-(dimethylamino)cyclohexyl)benzamide
|
|
Identifiers | |
CAS Number | 67579-24-2 ![]() |
ATC code | none |
PubChem | CID: 54753 |
ChemSpider | 49457 ![]() |
UNII | R8DWN01P1M ![]() |
ChEMBL | CHEMBL2110893 |
Synonyms | Bromadoline |
Chemical data | |
Formula | C15H21BrN2O |
Molecular mass | 325.244 g/mol |
|
|
|
|
(verify) |
Bromadoline (U-47931E)[1] is an opioid analgesic selective for the mu-opioid receptor[2] developed by the Upjohn company in the 1970s.[3] The drug has a potency lying between that of codeine and morphine being slightly stronger than pentazocine.[4] It is presumed that the (1R,2R) isomer is the active opioid, overlaying as it does with many other mu agonists.[5] Bromadoline is related to AH-7921 and U-47700.[6]
See also
References
- ↑ Lua error in package.lua at line 80: module 'strict' not found.
- ↑ Lua error in package.lua at line 80: module 'strict' not found.
- ↑ U.S. Patent 4,098,904
- ↑ Lua error in package.lua at line 80: module 'strict' not found.
- ↑ Lua error in package.lua at line 80: module 'strict' not found.
- ↑ Lua error in package.lua at line 80: module 'strict' not found.
<templatestyles src="Asbox/styles.css"></templatestyles>
Categories:
- Chemical articles having calculated molecular weight overwritten
- Infobox drug articles without a structure image
- Chemical pages without DrugBank identifier
- Articles without KEGG source
- Drugs not assigned an ATC code
- Drugs with no legal status
- Amines
- Benzamides
- Synthetic opioids
- Organobromides
- Mu-opioid agonists
- Nervous system drug stubs